MOTS-c — Mitochondrial-derived peptide. 16-residue sequence shown as a side-chain class strip (1 acidic, 4 basic, 4 aromatic, 1 polar, 6 nonpolar). Molecular weight ≈2174 g/mol.
Metabolic & Mitochondrial

MOTS-c

Mitochondrial-derived peptide

A mitochondrial-derived peptide studied in metabolic regulation and exercise research.

Also referenced as: Mitochondrial ORF of the 12S rRNA type-c, MOTSc

16 aa
For research and educational purposes only. This page is a factual research reference, not medical advice. Any dosing figures shown are amounts reported in the research literature, provided for educational context — not instructions or recommendations for human use.

Overview

MOTS-c (Mitochondrial ORF of the 12S rRNA type-c) is a 16-amino-acid mitochondrial-derived peptide encoded within the MT-RNR1 (12S rRNA) region of mitochondrial DNA. It was described in 2015 and is one of a small family of mitochondrial-derived peptides.

At a glance

ClassMitochondrial-derived peptide
CategoryMetabolic & Mitochondrial
SequenceMRWQEMGYIFYPRKLR
Chain length16 amino acids
Molecular weight~2174 g/mol
Typical formLyophilized powder
AliasesMitochondrial ORF of the 12S rRNA type-c, MOTSc
Use designationResearch / in-vitro only
Regulatory statusResearch-only / investigational. Not an approved drug; it is also a monitored substance in some anti-doping contexts. Educational and research use only, not medical advice.

What MOTS-c does

MOTS-c is a 16-amino-acid mitochondrial-derived peptide encoded within the mitochondrial 12S rRNA region, making it one of a small class of peptides written in the mitochondrial rather than nuclear genome. Its defining action in research is metabolic regulation through AMPK activation. Mechanistically, MOTS-c inhibits the folate cycle and its downstream de novo purine biosynthesis, causing accumulation of AICAR (an endogenous AMP mimetic), which in turn activates AMPK, the cell's master energy-sensing kinase. Skeletal muscle appears to be its primary target tissue. Under metabolic stress, MOTS-c also translocates to the nucleus and acts on stress-response gene expression, giving it a role as a signal that coordinates the cell's response to energy demand.

Downstream, AMPK activation by MOTS-c enhances insulin-independent glucose uptake, increases fatty-acid beta-oxidation, and improves whole-body insulin sensitivity. In mouse studies, MOTS-c administration prevented both age-dependent and high-fat-diet-induced insulin resistance and protected against diet-induced obesity, with roughly a 30% increase in the glucose infusion rate needed to maintain euglycemia during insulin clamps, a direct readout of improved insulin sensitivity. Because it reproduces several exercise-like metabolic adaptations, it is often described as an exercise-mimetic peptide. Human data are so far correlational rather than interventional: circulating MOTS-c levels have been found reduced in certain obese populations, and levels rise with exercise, but there are no completed controlled human efficacy trials, so the functional claims rest on animal and cell evidence.

Effects reported in research

  • Activates AMPK, the master cellular energy sensor, by inhibiting the folate cycle and raising endogenous AICAR (mechanistic/animal).
  • Enhances insulin-independent glucose uptake in skeletal muscle (its primary target tissue).
  • Improved whole-body insulin sensitivity (~30% higher glucose infusion rate in mouse insulin clamps).
  • Increased fatty-acid beta-oxidation, limiting fat accumulation in diet-induced obese mice.
  • Prevented age-dependent and high-fat-diet-induced insulin resistance in mouse models.
  • Protected against diet-induced obesity in rodents.
  • Translocates to the nucleus under metabolic stress to regulate stress-adaptive gene expression (cell-based data).
  • In humans, circulating levels are reduced in some obese populations and rise with exercise — associative only, no completed interventional efficacy trials.

Effects listed reflect findings reported in the research literature — many in animal or in-vitro models. Listing an effect is not a claim of efficacy or a therapeutic indication in humans.

Mechanism of action

MOTS-c is reported to regulate metabolic homeostasis, in part via activation of the AMPK pathway and modulation of the folate-methionine cycle and de novo purine biosynthesis. It has been described to translocate to the nucleus under metabolic stress and influence stress-response gene expression. Preclinical work links it to improved insulin sensitivity and glucose uptake in skeletal muscle; it is also described as exercise-responsive.

Mechanistic description reflects published research-literature understanding. Much peptide research is preclinical (in-vitro or animal-model); mechanism in humans may differ and is not established for many compounds.

What it's studied for

Research contexts in which MOTS-c appears in the literature. Listing a research area is not a claim of efficacy or a therapeutic indication.

Mitochondrial metabolism and AMPK signalingInsulin sensitivity and glucose homeostasis (preclinical)Exercise physiology / exercise-mimetic researchAging and metabolic-disease modelsNuclear stress-response gene regulation

Key characteristics

  • A genuine peptide encoded by mitochondrial DNA (mitochondrial-derived peptide)
  • 16 amino acids; sequence MRWQEMGYIFYPRKLR
  • Associated with AMPK activation and metabolic-stress adaptation in preclinical studies
  • Levels reported to change with exercise and age
  • Evidence is predominantly preclinical; not an approved therapeutic

Reported research dosing reference only

Educational reference, not dosing guidance. The figures below summarize amounts reported in published research and research-community protocols, provided for educational and research context only. They are not medical advice, not a recommendation, and not instructions for human use. MOTS-c is a research compound.

Reported research dosing comes from rodent studies rather than established human protocols. Published mouse work used systemic dosing on daily or intermittent schedules. These are figures reported for research context only, not dosing guidance for humans.

  • Rodent studies: reported at ~15 mg/kg/day for ~2 weeks
  • Rodent studies (intermittent): reported at ~15 mg/kg dosed ~3x/week
Reported frequencyReported as daily or intermittent (approximately 3x/week) in rodent studies
ReconstitutionLyophilized; typically reconstituted with bacteriostatic or sterile water

Human pharmacokinetics and dosing are not established; no completed published human trials. Reference figures only.

How it compares

Unlike the GH-derived fragments here, MOTS-c is endogenously encoded in the mitochondrial genome and acts as a broad metabolic regulator rather than a targeted lipolytic fragment.

Commonly studied alongside

Compounds frequently researched together with MOTS-c in the literature. Cross-referenced for research context — not a usage or combination recommendation.

Compare and calculate

Side-by-side pages for the pairings the literature already documents for MOTS-c, plus the unit-conversion reference for a reconstituted vial. Factual comparisons of documented characteristics — not a recommendation to combine or use any compound.

MOTS-c reconstitution calculator → Concentration, volume per measured amount and syringe units for a stated vial mass and diluent volume. A unit-conversion reference, not a dosing recommendation.

Handling & Stability

Lyophilized peptides are stored cold, protected from light, and reconstituted only at the time of intended in-vitro work.

  • Avoid repeated freeze-thaw cycles
  • Verify supplier lot and Certificate of Analysis
  • Follow institutional lab-safety protocols

Analytical & COA Concepts

Reputable research suppliers publish a third-party Certificate of Analysis per batch. Key analytical concepts referenced in COAs include:

Category Context

MOTS-c sits in the Metabolic & Mitochondrial area of the PeptiDex library.

Research Supplier Listing

Where researchers source MOTS-c

For researchers studying MOTS-c, third-party suppliers such as Practically Natty Peptides offer research-grade material, third-party tests every batch and provides Certificates of Analysis on request, and ship from the US.

View research-supplier listing →

Outbound link to a third-party research supplier. Inclusion does not constitute endorsement; all editorial content is developed independently.

Frequently asked questions

What is MOTS-c and where does it come from?

MOTS-c (Mitochondrial Open-reading-frame of the Twelve-S rRNA type-c) is a 16-amino-acid mitochondrial-derived peptide (MDP) encoded within the 12S rRNA region of mitochondrial DNA, rather than by the nuclear genome. First described in 2015, it is studied as a regulator of metabolic homeostasis. Its sequence and MDP origin make it structurally distinct from most catalog peptides.

What is MOTS-c studied for?

MOTS-c is studied in models of metabolic homeostasis, insulin sensitivity, exercise capacity, and aging. Research reported that MOTS-c levels rise with exercise and that exogenous MOTS-c improved glucose tolerance, insulin sensitivity, and running endurance in aged mice. It is thought to act partly via AMPK-linked metabolic signaling.

How is MOTS-c thought to work mechanistically?

MOTS-c is reported to translocate to the nucleus under metabolic stress and influence adaptive gene-expression programs, and it engages the AMPK pathway and folate/one-carbon metabolism to promote glucose uptake and fatty-acid oxidation. This positions it as a signaling peptide linking mitochondrial state to whole-body metabolism in preclinical models.

What does MOTS-c's pharmacokinetic profile imply for research design?

The pharmacokinetics of exogenous MOTS-c (bioavailability, distribution, half-life, clearance) are incompletely characterized in the literature, and no completed human clinical trials have been published. Rodent studies have used both daily and intermittent (e.g., 3x/week) dosing schedules, which reflects this uncertainty. Researchers should treat protocol parameters as provisional.

How should MOTS-c be reconstituted and stored?

MOTS-c is supplied as a white to off-white lyophilized powder, soluble in water, and is typically reconstituted with bacteriostatic or sterile water. Lyophilized peptide is stored refrigerated (2-8 C) or frozen for longer terms, with reconstituted solution kept refrigerated. A COA with HPLC purity and mass identity is standard.

Answers are educational summaries of research-literature context and do not constitute medical advice. See the Research Library, COA guide, and Storage & Handling guide for more.

References

Primary literature indexed in PubMed for MOTS-c. Listing a study records that it exists and is indexed — it is not a claim of efficacy, a therapeutic indication, or an endorsement of its conclusions. Much of this literature is preclinical (in-vitro or animal-model).

  1. The mitochondrial-derived peptide MOTS-c promotes metabolic homeostasis and reduces obesity and insulin resistance Cell Metab, 2015. PubMed 25738459
  2. The Mitochondrial-Encoded Peptide MOTS-c Translocates to the Nucleus to Regulate Nuclear Gene Expression in Response to Metabolic Stress Cell Metab, 2018. PubMed 29983246
  3. Mitochondria-derived peptide MOTS-c: effects and mechanisms related to stress, metabolism and aging J Transl Med, 2023. PubMed 36670507

Each reference was checked against its PubMed record on 2026-07-28: the PMID resolves and the title, journal and year match. Where no indexed literature exists for a compound, PeptiDex says so rather than substituting a citation about a different molecule. See the editorial policy.

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Further reading